Which of the following is described as a competitive benzodiazepine receptor antagonist?A.MidazolamB.FlumazenilC.KetamineD.Chlordiazepoxide

A competitive antagonist is a substance that:a.Binds to one receptor subtype as an agonist and to another as an antagonistb.Binds to the same receptor site and progressively inhibits the agonist responsec.Interacts with receptors and produces submaximal effectd.Binds to the nonspecific sites of tissueClear my choice

Which of the following is an antidepressant agent that selectively inhibits serotonin uptake with minimal effect on norepinephrine uptake?A.MaprotilineB.DespiramineC.FluoxetineD.Protriptyline

Differentiate betweenCompetitive and non-competitive inhibitors

Competitive antagonist differs from non-competitive in all the following except:a.It modifies drug potency, not efficacyb.Its effect can be reversed by increasing the dose of the agonistc.It reduces the maximal agonist response even with increasing the dosed.Shift the dose-response curve of the agonist to the right

...................inhibitors are molecules/compounds capable of binding to a region of the enzyme other than the active site.UncompetitiveNon-competitiveCompetitiveOver-competitive